Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50003348
LigandPNGBDBM50469638(NAPITANE)
Affinity DataKi:  0.428nMAssay Description:In vitro binding affinity at Alpha-2 adrenergic receptor in rat cortex by radioligand binding assay using [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50469636(CHEMBL25014)
Affinity DataKi:  0.5nMAssay Description:In vitro binding affinity at Alpha-2 adrenergic receptor in rat cortex by radioligand binding assay using [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50469635(Napitane)
Affinity DataKi:  0.708nMAssay Description:In vitro binding affinity at Alpha-2 adrenergic receptor in rat cortex by radioligand binding assay using [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50469635(Napitane)
Affinity DataKi:  0.708nMAssay Description:In vitro binding affinity at Alpha-2 adrenergic receptor in rat cortex by radioligand binding assay using [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50019848(2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1...)
Affinity DataKi:  1.70nMAssay Description:In vitro binding affinity at Alpha-2 adrenergic receptor in rat cortex by radioligand binding assay using [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50469637(CHEMBL285367)
Affinity DataKi:  2.10nMAssay Description:In vitro binding affinity at Alpha-2 adrenergic receptor in rat cortex by radioligand binding assay using [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50469634(CHEMBL433033)
Affinity DataKi:  4.60nMAssay Description:In vitro binding affinity at Alpha-2 adrenergic receptor in rat cortex by radioligand binding assay using [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50010859(CHEMBL11 | IMIPRAMINE HYDROCHLORIDE | IMIPRAMINE P...)
Affinity DataKi:  46nMAssay Description:In vitro binding affinity at Alpha-1 adrenergic receptor by radioligand binding assay using [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails ArticleDrugBank

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50469636(CHEMBL25014)
Affinity DataKi:  47nMAssay Description:In vitro binding affinity at Alpha-1 adrenergic receptor by radioligand binding assay using [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50469635(Napitane)
Affinity DataKi:  75.9nMAssay Description:In vitro binding affinity at Alpha-1 adrenergic receptor by radioligand binding assay using [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50469635(Napitane)
Affinity DataKi:  76nMAssay Description:In vitro binding affinity at Alpha-1 adrenergic receptor by radioligand binding assay using [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50469637(CHEMBL285367)
Affinity DataKi:  104nMAssay Description:In vitro binding affinity at Alpha-1 adrenergic receptor by radioligand binding assay using [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50469638(NAPITANE)
Affinity DataKi:  106nMAssay Description:In vitro binding affinity at Alpha-1 adrenergic receptor by radioligand binding assay using [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50469634(CHEMBL433033)
Affinity DataKi:  189nMAssay Description:In vitro binding affinity at Alpha-1 adrenergic receptor by radioligand binding assay using [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50010859(CHEMBL11 | IMIPRAMINE HYDROCHLORIDE | IMIPRAMINE P...)
Affinity DataKi:  255nMAssay Description:In vitro binding affinity at Alpha-2 adrenergic receptor in rat cortex by radioligand binding assay using [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50019848(2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1...)
Affinity DataKi:  403nMAssay Description:In vitro binding affinity at Alpha-1 adrenergic receptor by radioligand binding assay using [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails Article