Compile Data Set for Download or QSAR
maximum 50k data
Found 104 Enz. Inhib. hit(s) with all data for entry = 50004973
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50067424((S)-9-Methoxy-7-oxo-3b,4,5,6-tetrahydro-7H-2,6a,11...)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha5beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50067425((S)-9-Bromo-7-oxo-3b,4,5,6-tetrahydro-7H-2,6a,11b-...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha5beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
In DepthDetails Article
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50067420((S)-9-Ethynyl-7-oxo-3b,4,5,6-tetrahydro-7H-2,6a,11...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha5beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
In DepthDetails Article
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487291(CHEMBL2261918)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha5beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50487291(CHEMBL2261918)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha1beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487292(CHEMBL2261919)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha5beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50067439((S)-7-Oxo-9-trimethylsilanylethynyl-3b,4,5,6-tetra...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha5beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
In DepthDetails Article
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487295(CHEMBL2261922)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha5beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487299(CHEMBL2261632)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha5beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487296(CHEMBL2261633)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha5beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50487300(CHEMBL2261631)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha1beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487304(CHEMBL2261634)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha5beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487300(CHEMBL2261631)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha5beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487302(CHEMBL2261917)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha5beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA A receptor alpha-4/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487291(CHEMBL2261918)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-Ro 15-4513 from Homo sapiens (human) recombinant GABAA alpha4beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50487299(CHEMBL2261632)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha3beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487301(CHEMBL2261916)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha5beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50067425((S)-9-Bromo-7-oxo-3b,4,5,6-tetrahydro-7H-2,6a,11b-...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha3beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50487291(CHEMBL2261918)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha3beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50487302(CHEMBL2261917)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha1beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487291(CHEMBL2261918)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha2beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50067424((S)-9-Methoxy-7-oxo-3b,4,5,6-tetrahydro-7H-2,6a,11...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha3beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50487292(CHEMBL2261919)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha3beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA A receptor alpha-4/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487292(CHEMBL2261919)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-Ro 15-4513 from Homo sapiens (human) recombinant GABAA alpha4beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50067420((S)-9-Ethynyl-7-oxo-3b,4,5,6-tetrahydro-7H-2,6a,11...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha3beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
In DepthDetails Article
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50067424((S)-9-Methoxy-7-oxo-3b,4,5,6-tetrahydro-7H-2,6a,11...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha2beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50487301(CHEMBL2261916)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha1beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50067425((S)-9-Bromo-7-oxo-3b,4,5,6-tetrahydro-7H-2,6a,11b-...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha2beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
In DepthDetails Article
TargetGABA A receptor alpha-4/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487295(CHEMBL2261922)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-Ro 15-4513 from Homo sapiens (human) recombinant GABAA alpha4beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487299(CHEMBL2261632)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha2beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50487299(CHEMBL2261632)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha1beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487292(CHEMBL2261919)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha2beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487293(CHEMBL2261920)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha5beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50067420((S)-9-Ethynyl-7-oxo-3b,4,5,6-tetrahydro-7H-2,6a,11...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha2beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50487291(CHEMBL2261918)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]-Ro 15-4513 from Homo sapiens (human) recombinant GABAA alpha6beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50067425((S)-9-Bromo-7-oxo-3b,4,5,6-tetrahydro-7H-2,6a,11b-...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]-Ro 15-4513 from Homo sapiens (human) recombinant GABAA alpha6beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50067425((S)-9-Bromo-7-oxo-3b,4,5,6-tetrahydro-7H-2,6a,11b-...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha1beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50067424((S)-9-Methoxy-7-oxo-3b,4,5,6-tetrahydro-7H-2,6a,11...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha1beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50487295(CHEMBL2261922)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha3beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50487292(CHEMBL2261919)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha1beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA A receptor alpha-4/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487300(CHEMBL2261631)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]-Ro 15-4513 from Homo sapiens (human) recombinant GABAA alpha4beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50487300(CHEMBL2261631)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha3beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487300(CHEMBL2261631)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha2beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487296(CHEMBL2261633)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha2beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))TBA
LigandPNGBDBM50487298(CHEMBL2261915)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha5beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50487292(CHEMBL2261919)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]-Ro 15-4513 from Homo sapiens (human) recombinant GABAA alpha6beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50067420((S)-9-Ethynyl-7-oxo-3b,4,5,6-tetrahydro-7H-2,6a,11...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha1beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50487301(CHEMBL2261916)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha3beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50487296(CHEMBL2261633)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]-Ro 15-1788 from Homo sapiens (human) recombinant GABAA alpha3beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM50487295(CHEMBL2261922)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]-Ro 15-4513 from Homo sapiens (human) recombinant GABAA alpha6beta3gamma2 receptor expressed in Ltk- cells after 1 hr by liquid s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
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