Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50005106
TargetRyanodine receptor 1(Oryctolagus cuniculus)
University of California

Curated by ChEMBL
LigandPNGBDBM50044994(2,6,9,11,13,14-hexahydroxy-11-isopropyl-3,7,10-tri...)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]ryanodine from Ca2+-ryanodine receptor in Oryctolagus cuniculus (rabbit) skeletal muscle sarcoplasmic reticulum after 2 hr by com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRyanodine receptor 3(Mus musculus)
University of California

Curated by ChEMBL
LigandPNGBDBM50044994(2,6,9,11,13,14-hexahydroxy-11-isopropyl-3,7,10-tri...)
Affinity DataIC50:  3.30nMAssay Description:Binding affinity to ryanodine receptor in Mus musculus albino Swiss-Webster (mouse) brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRyanodine receptor 1(Oryctolagus cuniculus)
University of California

Curated by ChEMBL
LigandPNGBDBM50044994(2,6,9,11,13,14-hexahydroxy-11-isopropyl-3,7,10-tri...)
Affinity DataIC50:  3.5nMAssay Description:Displacement of [3H]ryanodine from Ca2+-ryanodine receptor in Oryctolagus cuniculus (rabbit) skeletal muscle sarcoplasmic reticulum after 1 hr by com...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed