Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50005430
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50491996(CHEMBL2391644)
Affinity DataIC50:  18nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50223136(CHEMBL249360 | N-((R)-1-((R)-7-chloro-1-isopropyl-...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50491995(CHEMBL2391645)
Affinity DataIC50:  34nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50216671(CHEMBL247828 | tert-butyl (R)-1-((R)-1-isopropyl-2...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50491993(CHEMBL2391648)
Affinity DataIC50:  57nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50491998(CHEMBL2391649)
Affinity DataIC50:  67nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50491997(CHEMBL2391643)
Affinity DataIC50:  70nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50491990(CHEMBL2391790)
Affinity DataIC50:  85nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50492007(CHEMBL2391792)
Affinity DataIC50:  101nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50492005(CHEMBL2391788)
Affinity DataIC50:  103nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50492002(CHEMBL2391785)
Affinity DataIC50:  103nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50223137(CHEMBL251346 | tert-butyl (R)-1-((R)-7-chloro-1-is...)
Affinity DataIC50:  108nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50491989(CHEMBL2391791)
Affinity DataIC50:  117nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50491988(CHEMBL2391642)
Affinity DataIC50:  131nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50492001(CHEMBL2391789)
Affinity DataIC50:  137nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50492004(CHEMBL2391646)
Affinity DataIC50:  181nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50492000(CHEMBL2391787)
Affinity DataIC50:  229nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50492003(CHEMBL2391650)
Affinity DataIC50:  254nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50491999(CHEMBL2391784)
Affinity DataIC50:  260nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50492006(CHEMBL2391783)
Affinity DataIC50:  264nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50491992(CHEMBL2391782)
Affinity DataIC50:  359nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50491991(CHEMBL2391786)
Affinity DataIC50:  443nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50491994(CHEMBL2391647)
Affinity DataIC50:  494nMAssay Description:Inhibition of human NaV1.7 channel expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed