Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50007645
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511159(CHEMBL4550946)
Affinity DataIC50:  13nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511162(CHEMBL4575812)
Affinity DataIC50:  14nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511154(CHEMBL4442374)
Affinity DataIC50:  19nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511152(CHEMBL4474836)
Affinity DataIC50:  25nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)
Affinity DataIC50:  27nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511155(CHEMBL4456985)
Affinity DataIC50:  27nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511150(CHEMBL4440790)
Affinity DataIC50:  39nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511164(CHEMBL4514653)
Affinity DataIC50:  56nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511156(CHEMBL4521356)
Affinity DataIC50:  64nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511161(CHEMBL4579529)
Affinity DataIC50:  74nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511165(CHEMBL4563765)
Affinity DataIC50:  84nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511158(CHEMBL4437998)
Affinity DataIC50:  97nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511157(CHEMBL4552025)
Affinity DataIC50:  98nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511160(CHEMBL4513287)
Affinity DataIC50:  112nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511153(CHEMBL4564623)
Affinity DataIC50:  139nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50379523(CHEMBL2012558)
Affinity DataIC50:  152nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511151(CHEMBL4483653)
Affinity DataIC50:  168nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511147(CHEMBL4476003)
Affinity DataIC50:  168nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511149(CHEMBL4438785)
Affinity DataIC50:  215nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511148(CHEMBL4539999)
Affinity DataIC50:  950nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50511163(CHEMBL4528315)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) by FRET-based Lantha-screen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed