BindingDB PrimarySearch_ki

Found 128 Enz. Inhib. hit(s) with all data for entry = 50009645

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530623(CHEMBL4521381)

IC50: 0.0430nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair

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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530623(CHEMBL4521381)

IC50: 0.0430nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50468247(HM 781-36B | HM-781-36B | NOV-120101 | Poziotinib ...)

IC50: 0.0780nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50468247(HM 781-36B | HM-781-36B | NOV-120101 | Poziotinib ...)

IC50: 0.0780nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530623(CHEMBL4521381)

IC50: 0.133nMAssay Description:Inhibition of GST-tagged human EGFR D770_N771insNPG mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent k...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530623(CHEMBL4521381)

IC50: 0.133nMAssay Description:Inhibition of GST-tagged human EGFR D770_N771insNPG mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent k...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530618(CHEMBL4559807)

IC50: 0.145nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530618(CHEMBL4559807)

IC50: 0.145nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530622(CHEMBL4514452)

IC50: 0.214nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair

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Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530622(CHEMBL4514452)

IC50: 0.214nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50468247(HM 781-36B | HM-781-36B | NOV-120101 | Poziotinib ...)

IC50: 0.218nMAssay Description:Inhibition of GST-tagged human EGFR D770_N771insNPG mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent k...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50468247(HM 781-36B | HM-781-36B | NOV-120101 | Poziotinib ...)

IC50: 0.218nMAssay Description:Inhibition of GST-tagged human EGFR D770_N771insNPG mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent k...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50029668(AZD-9291 | Osimertinib | US10085983, Compound AZD-...)

IC50: 0.421nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair

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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50029668(AZD-9291 | Osimertinib | US10085983, Compound AZD-...)

IC50: 0.421nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair

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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530618(CHEMBL4559807)

IC50: 0.636nMAssay Description:Inhibition of GST-tagged human EGFR D770_N771insNPG mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent k...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530618(CHEMBL4559807)

IC50: 0.636nMAssay Description:Inhibition of GST-tagged human EGFR D770_N771insNPG mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent k...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50029668(AZD-9291 | Osimertinib | US10085983, Compound AZD-...)

IC50: 0.950nMAssay Description:Inhibition of GST-tagged human EGFR D770_N771insNPG mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent k...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50029668(AZD-9291 | Osimertinib | US10085983, Compound AZD-...)

IC50: 0.950nMAssay Description:Inhibition of GST-tagged human EGFR D770_N771insNPG mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent k...More data for this Ligand-Target Pair

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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530615(CHEMBL4534719)

IC50: 1.20nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530615(CHEMBL4534719)

IC50: 1.20nMAssay Description:Inhibition of GST-tagged human EGFR A763_Y764insFHEA mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530622(CHEMBL4514452)

IC50: 1.5nMAssay Description:Inhibition of GST-tagged human EGFR D770_N771insNPG mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent k...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530622(CHEMBL4514452)

IC50: 1.5nMAssay Description:Inhibition of GST-tagged human EGFR D770_N771insNPG mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent k...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530632(CHEMBL4458437)

IC50: 13nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530632(CHEMBL4458437)

IC50: 13nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530624(CHEMBL4463012)

IC50: 14nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50322823((S)-N-(4-(3-chloro-4-fluorophenylamino)-7-(tetrahy...)

IC50: 14nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530624(CHEMBL4463012)

IC50: 14nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50322823((S)-N-(4-(3-chloro-4-fluorophenylamino)-7-(tetrahy...)

IC50: 14nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530623(CHEMBL4521381)

IC50: 15nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530623(CHEMBL4521381)

IC50: 15nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530615(CHEMBL4534719)

IC50: 18nMAssay Description:Inhibition of GST-tagged human EGFR D770_N771insNPG mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent k...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530615(CHEMBL4534719)

IC50: 18nMAssay Description:Inhibition of GST-tagged human EGFR D770_N771insNPG mutant using poly(Glu, Tyr) 4:1 substrate incubated for 120 mins by kinase-Glo plus luminescent k...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530631(CHEMBL4583178)

IC50: 19nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530631(CHEMBL4583178)

IC50: 19nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50322822((S)-N-(3-(4-(2-hydroxy-1-phenylethylamino)-6-pheny...)

IC50: 20nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50322822((S)-N-(3-(4-(2-hydroxy-1-phenylethylamino)-6-pheny...)

IC50: 20nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50322823((S)-N-(4-(3-chloro-4-fluorophenylamino)-7-(tetrahy...)

IC50: 22nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50322823((S)-N-(4-(3-chloro-4-fluorophenylamino)-7-(tetrahy...)

IC50: 22nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530618(CHEMBL4559807)

IC50: 24nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530618(CHEMBL4559807)

IC50: 24nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50322822((S)-N-(3-(4-(2-hydroxy-1-phenylethylamino)-6-pheny...)

IC50: 27nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50322822((S)-N-(3-(4-(2-hydroxy-1-phenylethylamino)-6-pheny...)

IC50: 27nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)

IC50: 29nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)

IC50: 29nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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PDB

3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530623(CHEMBL4521381)

IC50: 48nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530623(CHEMBL4521381)

IC50: 48nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain I858R/T790M mutant (696 to 1022 residues) using EGFR L858R/T790M substrate peptide incubated for 12...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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3D Structure (crystal)

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530635(CHEMBL4448691)

IC50: 62nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530635(CHEMBL4448691)

IC50: 62nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530627(CHEMBL4456359)

IC50: 64nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Epidermal growth factor receptor(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL

PNG

BDBM50530627(CHEMBL4456359)

IC50: 64nMAssay Description:Inhibition of GST-tagged human EGFR kinase domain (696 to 1022 residues) using poly(Glu, Tyr) 4:1 substrate incubated for 60 mins by kinase-Glo plus ...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

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