TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:In vitro inhibitory concentration against human mitogen-activated protein kinase-1 (MEK-1) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:In vitro inhibitory concentration against checkpoint kinase 2 (Chk2) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:In vitro inhibitory concentration against human casein kinase 1 delta (CK1 delta) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:In vitro inhibitory concentration against checkpoint kinase 2 (Chk2) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 89nMAssay Description:In vitro inhibitory concentration against human mitogen-activated protein kinase-1 (MEK-1) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 183nMAssay Description:In vitro inhibitory concentration against checkpoint kinase 2 (Chk2) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 237nMAssay Description:In vitro inhibitory concentration against checkpoint kinase 1 (Chk1) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:In vitro inhibitory concentration against human protein kinase C alpha (PKCa) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 725nMAssay Description:In vitro inhibitory concentration against checkpoint kinase 1 (Chk1) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 824nMAssay Description:In vitro inhibitory concentration against human mitogen-activated protein kinase-1 (MEK-1) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro inhibitory concentration against human protein kinase C beta-2 (PKCbetaII) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.35E+3nMAssay Description:In vitro inhibitory concentration against human casein kinase 1 delta (CK1 delta) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 1.95E+3nMAssay Description:In vitro inhibitory concentration against checkpoint kinase 1 (Chk1) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.54E+3nMAssay Description:In vitro inhibitory concentration against human protein kinase C alpha (PKCa) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.38E+3nMAssay Description:In vitro inhibitory concentration against human protein kinase C beta-2 (PKCbetaII) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:In vitro inhibitory concentration against human casein kinase 2 (CK2) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Michigan State University
Curated by ChEMBL
Michigan State University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibitory concentration against human casein kinase 2 (CK2) by using [gamma-33P]-ATP] as radioligandMore data for this Ligand-Target Pair