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Found 20 Enz. Inhib. hit(s) with all data for entry = 50018523
TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50443101(Cariprazine | RGH-188)
Affinity DataKi:  0.0850nMAssay Description:Partial agonist activity at human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  0.340nMAssay Description:Partial agonist activity at human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  0.800nMAssay Description:Partial agonist activity at human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50609164(CHEMBL5289063)
Affinity DataKi:  3.40nMAssay Description:Partial agonist activity at human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50518031(CHEMBL4445841)
Affinity DataKi:  12nMAssay Description:Partial agonist activity at human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609163(CHEMBL5272965)
Affinity DataKi:  27nMAssay Description:Partial agonist activity at human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  44nMAssay Description:Partial agonist activity at human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
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TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50518031(CHEMBL4445841)
Affinity DataKi:  79nMAssay Description:Partial agonist activity at human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50609163(CHEMBL5272965)
Affinity DataKi:  139nMAssay Description:Partial agonist activity at human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50518031(CHEMBL4445841)
Affinity DataKi:  170nMAssay Description:Partial agonist activity at human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609164(CHEMBL5289063)
Affinity DataKi:  190nMAssay Description:Partial agonist activity at human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50443101(Cariprazine | RGH-188)
Affinity DataEC50:  0.180nMAssay Description:Partial agonist activity at human D2 receptor assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609163(CHEMBL5272965)
Affinity DataEC50:  62nMAssay Description:Partial agonist activity at human D2 receptor assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609165(CHEMBL5266559)
Affinity DataEC50:  260nMAssay Description:Partial agonist activity at human D2 receptor expressed in CHO-K1 cells assessed as forskolin-stimulated cAMP production incubated for 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataEC50:  2.40nMAssay Description:Partial agonist activity at human D2 receptor assessed as beta arrestin-2 recruitmentMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609163(CHEMBL5272965)
Affinity DataEC50:  840nMAssay Description:Partial agonist activity at human D2 receptor assessed as beta arrestin-2 recruitmentMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609164(CHEMBL5289063)
Affinity DataEC50:  250nMAssay Description:Partial agonist activity at human D2 receptor assessed as beta arrestin-2 recruitmentMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50518031(CHEMBL4445841)
Affinity DataEC50:  6.30nMAssay Description:Partial agonist activity at D2 receptor (unknown origin) assessed as beta arrestin-2 recruitmentMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataEC50:  38nMAssay Description:Partial agonist activity at human D2 receptor assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609164(CHEMBL5289063)
Affinity DataEC50:  90nMAssay Description:Partial agonist activity at human D2 receptor assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed