Affinity DataKi: 0.0850nMAssay Description:Partial agonist activity at human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.340nMAssay Description:Partial agonist activity at human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Partial agonist activity at human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Partial agonist activity at human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Partial agonist activity at human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Partial agonist activity at human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Partial agonist activity at human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Partial agonist activity at human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 139nMAssay Description:Partial agonist activity at human D3 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Partial agonist activity at human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Partial agonist activity at human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataEC50: 0.180nMAssay Description:Partial agonist activity at human D2 receptor assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 62nMAssay Description:Partial agonist activity at human D2 receptor assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 260nMAssay Description:Partial agonist activity at human D2 receptor expressed in CHO-K1 cells assessed as forskolin-stimulated cAMP production incubated for 60 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.40nMAssay Description:Partial agonist activity at human D2 receptor assessed as beta arrestin-2 recruitmentMore data for this Ligand-Target Pair
Affinity DataEC50: 840nMAssay Description:Partial agonist activity at human D2 receptor assessed as beta arrestin-2 recruitmentMore data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Partial agonist activity at human D2 receptor assessed as beta arrestin-2 recruitmentMore data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:Partial agonist activity at D2 receptor (unknown origin) assessed as beta arrestin-2 recruitmentMore data for this Ligand-Target Pair
Affinity DataEC50: 38nMAssay Description:Partial agonist activity at human D2 receptor assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 90nMAssay Description:Partial agonist activity at human D2 receptor assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair