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Found 30 Enz. Inhib. hit(s) with all data for entry = 50018610
LigandPNGBDBM50610280(CHEMBL5267183)
Affinity DataEC50:  874nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50541163(CHEMBL4639024)
Affinity DataEC50:  880nMAssay Description:Induction of HMGCR degradation (unknown origin)More data for this Ligand-Target Pair
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LigandPNGBDBM50610282(CHEMBL5277972)
Affinity DataEC50:  722nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610283(CHEMBL5268887)
Affinity DataEC50:  336nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610284(CHEMBL5276325)
Affinity DataEC50:  152nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610285(CHEMBL5275821)
Affinity DataEC50:  351nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610286(CHEMBL5275694)
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610287(CHEMBL5276525)
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610288(CHEMBL5289887)
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610289(CHEMBL5282835)
Affinity DataEC50:  832nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610290(CHEMBL5271654)
Affinity DataEC50:  337nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610291(CHEMBL5290557)
Affinity DataEC50:  450nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610292(CHEMBL5288010)
Affinity DataEC50:  693nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610293(CHEMBL5266489)
Affinity DataEC50:  1.45E+3nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50559939(CHEMBL4756373)
Affinity DataEC50:  132nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610294(CHEMBL5266129)
Affinity DataEC50:  598nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610295(CHEMBL5290996)
Affinity DataEC50:  2.26E+3nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610296(CHEMBL5282672)
Affinity DataEC50:  311nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610297(CHEMBL5269334)
Affinity DataEC50:  389nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610298(CHEMBL5283544)
Affinity DataEC50:  492nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610299(CHEMBL5267256)
Affinity DataEC50:  98nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610300(CHEMBL5288099)
Affinity DataEC50:  102nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610301(CHEMBL5269782)
Affinity DataEC50:  98nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610302(CHEMBL5277572)
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610303(CHEMBL5280701)
Affinity DataEC50: >1.00E+4nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610304(CHEMBL5266062)
Affinity DataEC50:  356nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50610305(CHEMBL5284059)
Affinity DataEC50:  84nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50605021(CHEMBL5177065)
Affinity DataEC50:  390nMAssay Description:Induction of HMGCR degradation in CHO-7 cells incubated for 16 hrs by immunoblotting assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50559942(CHEMBL4760244)
Affinity DataEC50:  1.10E+3nMAssay Description:Induction of HMGCR degradation in human HepG2 cells incubated for 3 hrs by densitometric analysisMore data for this Ligand-Target Pair
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LigandPNGBDBM50610281(CHEMBL5275570)
Affinity DataEC50:  990nMAssay Description:Induction of HMGCR degradation in HEK293 cells incubated for 4 hrs by luciferase based assayMore data for this Ligand-Target Pair
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