Compile Data Set for Download or QSAR
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Found 38 Enz. Inhib. hit(s) with all data for entry = 50018985
TargetBifunctional glutamate/proline--tRNA ligase(Homo sapiens (Human))TBA
LigandPNGBDBM50614449(CHEMBL1163086)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human Prolyl-tRNA synthetaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetProline--tRNA ligase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50614449(CHEMBL1163086)
Affinity DataKi:  4.30nMAssay Description:Binding affinity to Escherichia coli K12 Prolyl-tRNA synthetaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetBifunctional glutamate/proline--tRNA ligase(Homo sapiens (Human))TBA
LigandPNGBDBM50614450(CHEMBL5279127)
Affinity DataKi:  85nMAssay Description:Binding affinity to human Prolyl-tRNA synthetaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50614446(CHEMBL5283680)
Affinity DataKi:  232nMAssay Description:Binding affinity to ADK (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlutamine--tRNA ligase(Escherichia coli)TBA
LigandPNGBDBM50614451(CHEMBL5291357)
Affinity DataKi:  280nMAssay Description:Binding affinity to Escherichia coli K12 glutaminyl-tRNA synthetase assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProline--tRNA ligase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50614450(CHEMBL5279127)
Affinity DataKi:  490nMAssay Description:Binding affinity to Escherichia coli K12 Prolyl-tRNA synthetaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))TBA
LigandPNGBDBM50614428(CHEMBL5283919)
Affinity DataKi:  690nMAssay Description:Binding affinity to human HGPRT assessed as inhibition of constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50614445(CHEMBL5282738)
Affinity DataIC50:  10nMAssay Description:Inhibition of MraY in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50614431(CHEMBL5289236)
Affinity DataIC50:  12nMAssay Description:Antimicrobial activity against Enterococcus faecalis ATCC 29212 assessed as microbial growth inhibitionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMethionine--tRNA ligase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50614447(CHEMBL5287030)
Affinity DataIC50:  14nMAssay Description:Inhibition of Escherichia coli K12 methionyl tRNA synthetaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Staphylococcus aureus (strain MRSA252))TBA
LigandPNGBDBM50614429(CHEMBL5265940)
Affinity DataIC50:  17nMAssay Description:Inhibition of Staphylococcus aureus MraYMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50614433(CHEMBL5272467)
Affinity DataIC50:  22nMAssay Description:Inhibition of Bacillus subtilis MraYMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Staphylococcus aureus (strain MRSA252))TBA
LigandPNGBDBM50614430(CHEMBL5277590)
Affinity DataIC50:  27nMAssay Description:Inhibition of Staphylococcus aureus MraYMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM50614432(CHEMBL5271984)
Affinity DataIC50:  42nMAssay Description:Inhibition of Bacillus subtilis MraYMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50614442(CHEMBL5278937)
Affinity DataIC50:  58nMAssay Description:Inhibition of MraY in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAlpha-1-antichymotrypsin(Homo sapiens)TBA
LigandPNGBDBM50614452(CHEMBL5291453)
Affinity DataIC50:  145nMAssay Description:Inhibition of ACT (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50614440(CHEMBL5281271)
Affinity DataIC50:  330nMAssay Description:Inhibition of MraY in Escherichia coli K12More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50614439(CHEMBL5276993)
Affinity DataIC50:  330nMAssay Description:Inhibition of MraY in Escherichia coli K12More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50614434(CHEMBL5288850)
Affinity DataIC50:  330nMAssay Description:Inhibition of MraY in Escherichia coli K12More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50614436(CHEMBL5267618)
Affinity DataIC50:  330nMAssay Description:Inhibition of MraY in Escherichia coli K12More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50614437(CHEMBL5275061)
Affinity DataIC50:  330nMAssay Description:Inhibition of MraY in Escherichia coli K12More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50614444(CHEMBL5284675)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of MraY in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMethionine--tRNA ligase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50614448(CHEMBL1161585)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of Escherichia coli K12 methionyl tRNA synthetaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50526659(CHEMBL4441639)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of MraY in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50526658(CHEMBL4555507)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of MraY in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50614443(CHEMBL5278566)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of MraY in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50526646(CHEMBL4452848)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of MraY in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50614441(CHEMBL5270917)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of MraY in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50526663(CHEMBL4521972)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of MraY in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50526668(CHEMBL4455936)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of MraY in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50526636(CHEMBL4577355)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of MraY in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50614438(CHEMBL149413)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of MraY in Escherichia coli K12More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50614435(CHEMBL151287)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of MraY in Escherichia coli K12More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50091506(1-[(2R,3R,4S,5R)-5-((2R,3R,4S,5R)-5-Aminomethyl-3,...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of MraY in Escherichia coli K12More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50097053(1-[5-[3,4-dihydroxy-5-iminomethylaminomethyl-(2R,3...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of MraY in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50097055(1-[5-[3,4-dihydroxy-5-methylaminomethyl-(2R,3R,4R,...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of MraY in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50097058(1-[5-[5-amino(imino)methylaminomethyl-3,4-dihydrox...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of MraY in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))TBA
LigandPNGBDBM50091506(1-[(2R,3R,4S,5R)-5-((2R,3R,4S,5R)-5-Aminomethyl-3,...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of MraY in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails PubMed