Affinity DataKi: 112nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 114nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 202nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 213nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 380nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 469nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 805nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 991nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.02E+3nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.47E+3nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >1.70E+3nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.75E+3nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >2.16E+3nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >2.37E+3nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >2.78E+3nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >3.23E+3nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >3.31E+3nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >3.80E+3nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >4.50E+3nMAssay Description:Inhibition of adrenergic alpha2A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 31nMAssay Description:Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >7.00E+3nMAssay Description:Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 51nMAssay Description:Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 729nMAssay Description:Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 0.400nMAssay Description:Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >6.50E+3nMAssay Description:Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 391nMAssay Description:Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >1.40E+3nMAssay Description:Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 146nMAssay Description:Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 92nMAssay Description:Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >3.57E+3nMAssay Description:Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >3.40E+3nMAssay Description:Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human adrenergic alpha1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: >2.60E+3nMAssay Description:Agonist activity at human adrenergic alpha1D receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 62nMAssay Description:Agonist activity at human adrenergic alpha1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair