Affinity DataKi: 0.5nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11.9nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11.9nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 16.6nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 24.6nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of muscarinic M1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 92nMAssay Description:Antagonist activity at histamine H1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Inhibition of muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 340nMAssay Description:Inhibition of muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 430nMAssay Description:Inhibition of muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 480nMAssay Description:Inhibition of muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 930nMAssay Description:Inhibition of muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 2.60E+3nMAssay Description:Displacement of [3H]dofetolide from human ErgMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 2.80E+3nMAssay Description:Inhibition of muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 2.90E+3nMAssay Description:Inhibition of muscarinic M1 receptorMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]dofetolide from human ErgMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]dofetolide from human ErgMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]dofetolide from human ErgMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]dofetolide from human ErgMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]dofetolide from human ErgMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]dofetolide from human ErgMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]dofetolide from human ErgMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]dofetolide from human ErgMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]dofetolide from human ErgMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]dofetolide from human ErgMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataKi: 3.90E+3nMAssay Description:Displacement of [3H]dofetolide from human ErgMore data for this Ligand-Target Pair