Compile Data Set for Download or QSAR
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Found 13 Enz. Inhib. hit(s) with all data for entry = 50035892
TargetMu-type opioid receptor(CALF)
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50013761((R)-1-(3-cyclopropylmethyl-11,15-dimethoxy-13-oxa-...)
Affinity DataIC50:  0.320nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50013388(6-Ethyl-3-(1-hydroxy-cyclopropylmethyl)-11,11-dime...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50406411(CHEMBL2021332)
Affinity DataIC50:  0.760nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50013764(5-(3-cyclopropylmethyl-11-hydroxy-15-methoxy-13-ox...)
Affinity DataIC50:  1nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50001714(2-[3-cyclopropylmethyl-11-hydroxy-15-methoxy-(1S,2...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataIC50:  5nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50013763((S)-19-(1-isothiocyanatoethyl)-15-methoxy-3-methyl...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50013768(3-O-(tert-Butyldimethylsilyl)-6,14-endo-etheno-7al...)
Affinity DataIC50:  34nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50406413(CHEMBL2021335)
Affinity DataIC50:  63nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50013769((S)-1-(3-cyclopropylmethyl-11,15-dimethoxy-13-oxa-...)
Affinity DataIC50:  171nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50013766((S)-1-(11,15-dimethoxy-3-methyl-13-oxa-3-azahexacy...)
Affinity DataIC50:  323nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50406412(CHEMBL2021333)
Affinity DataIC50:  434nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(CALF)
University Of Washington

Curated by ChEMBL
LigandPNGBDBM50013760((R)-1-(11,15-dimethoxy-3-methyl-13-oxa-3-azahexacy...)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of 0.5 nM [3H]- Bremazocine binding to Opioid receptor mu 1 of bovine striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed