Compile Data Set for Download or QSAR
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Found 9 Enz. Inhib. hit(s) with all data for entry = 50037618
TargetAromatase(Homo sapiens (Human))
University Of Oporto

Curated by ChEMBL
LigandPNGBDBM50174541((3R,4S,5R,10R,13S)-10,13-Dimethyl-hexadecahydro-20...)
Affinity DataKi:  38nMAssay Description:Inhibition constant against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Oporto

Curated by ChEMBL
LigandPNGBDBM50174544((5S,10S,13S)-10,13-Dimethyl-1,2,5,6,7,8,9,10,11,12...)
Affinity DataKi:  50nMAssay Description:Inhibition constant against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Oporto

Curated by ChEMBL
LigandPNGBDBM50174543((3R,5R,10R,13S)-3-Hydroxy-10,13-dimethyl-tetradeca...)
Affinity DataKi:  147nMAssay Description:Inhibition constant against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Oporto

Curated by ChEMBL
LigandPNGBDBM50174542((10aR,12aS)-7-Hydroxy-10a,12a-dimethyl-3,4,4a,5,6,...)
Affinity DataKi:  660nMAssay Description:Inhibition constant against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Oporto

Curated by ChEMBL
LigandPNGBDBM50240798((8R,9S,10R,13S,14S)-4-Hydroxy-10,13-dimethyl-1,6,7...)
Affinity DataIC50:  42nMAssay Description:Inhibitory concentration against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Oporto

Curated by ChEMBL
LigandPNGBDBM50174541((3R,4S,5R,10R,13S)-10,13-Dimethyl-hexadecahydro-20...)
Affinity DataIC50:  145nMAssay Description:Inhibitory concentration against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Oporto

Curated by ChEMBL
LigandPNGBDBM50174544((5S,10S,13S)-10,13-Dimethyl-1,2,5,6,7,8,9,10,11,12...)
Affinity DataIC50:  225nMAssay Description:Inhibitory concentration against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Oporto

Curated by ChEMBL
LigandPNGBDBM50174543((3R,5R,10R,13S)-3-Hydroxy-10,13-dimethyl-tetradeca...)
Affinity DataIC50:  670nMAssay Description:Inhibitory concentration against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Oporto

Curated by ChEMBL
LigandPNGBDBM50174542((10aR,12aS)-7-Hydroxy-10a,12a-dimethyl-3,4,4a,5,6,...)
Affinity DataIC50:  1.85E+3nMAssay Description:Inhibitory concentration against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed