Report error Found 67 Enz. Inhib. hit(s) with all data for entry = 50046357
Affinity DataIC50: 0.740nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of IRAK4-dependent TLR4 signaling in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of LP...More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibition of IRAK4-dependent TLR4 signaling in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of LP...More data for this Ligand-Target Pair
Affinity DataIC50: 87nMAssay Description:Inhibition of IRAK4-dependent TLR4 signaling in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of LP...More data for this Ligand-Target Pair
Affinity DataIC50: 89nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 94nMAssay Description:Inhibition of IRAK4-dependent TLR4 signaling in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of LP...More data for this Ligand-Target Pair
Affinity DataIC50: 94nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 113nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 155nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 204nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 216nMAssay Description:Inhibition of IRAK4-dependent TLR4 signaling in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of LP...More data for this Ligand-Target Pair
Affinity DataIC50: 341nMAssay Description:Inhibition of IRAK4-dependent TLR4 signaling in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of LP...More data for this Ligand-Target Pair
Affinity DataIC50: 373nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 647nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 852nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 932nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.45E+3nMAssay Description:Inhibition of IRAK4-dependent TLR4 signaling in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of LP...More data for this Ligand-Target Pair
Affinity DataIC50: 6.01E+3nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 9.51E+3nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human IRAK4 (unknown origin)More data for this Ligand-Target Pair
TargetTumor necrosis factor receptor superfamily member 1A(Human)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: >3.10E+4nMAssay Description:Inhibition of TNFR in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of TNFalpha-induced TNFR activa...More data for this Ligand-Target Pair
TargetTumor necrosis factor receptor superfamily member 1A(Human)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: >3.10E+4nMAssay Description:Inhibition of TNFR in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of TNFalpha-induced TNFR activa...More data for this Ligand-Target Pair
TargetTumor necrosis factor receptor superfamily member 1A(Human)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: >3.10E+4nMAssay Description:Inhibition of TNFR in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of TNFalpha-induced TNFR activa...More data for this Ligand-Target Pair
TargetTumor necrosis factor receptor superfamily member 1A(Human)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: >3.10E+4nMAssay Description:Inhibition of TNFR in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of TNFalpha-induced TNFR activa...More data for this Ligand-Target Pair
TargetTumor necrosis factor receptor superfamily member 1A(Human)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: >3.10E+4nMAssay Description:Inhibition of TNFR in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of TNFalpha-induced TNFR activa...More data for this Ligand-Target Pair
TargetTumor necrosis factor receptor superfamily member 1A(Human)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: >3.10E+4nMAssay Description:Inhibition of TNFR in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of TNFalpha-induced TNFR activa...More data for this Ligand-Target Pair
TargetTumor necrosis factor receptor superfamily member 1A(Human)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: >3.10E+4nMAssay Description:Inhibition of TNFR in human THP1-XBlue cells containing NF-kappaB-inducible SEAP reporter gene assessed as inhibition of TNFalpha-induced TNFR activa...More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair