Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50048245
TargetREST corepressor 1 [4-485](Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50158884(CHEMBL3785550)
Affinity DataKi:  140nMAssay Description:Inhibition of recombinant human His-tagged LSD1 (171 to 836 residues)/GST-tagged CoREST (308 to 440 residues) complex using H3K4 peptide substrate by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50210048(CHEMBL3884919)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of human LSD1 assessed as reduction in H2O2 production using H3K4me2 (1 to 20 residues) peptide as substrate preincubated for 10 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50158884(CHEMBL3785550)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of human LSD1 assessed as reduction in H2O2 production using H3K4me2 (1 to 20 residues) peptide as substrate preincubated for 10 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50210048(CHEMBL3884919)
Affinity DataKi:  3.70E+4nMAssay Description:Inhibition of human LSD1 assessed as reduction in H2O2 production using H3K4me2 (1 to 20 residues) peptide as substrate preincubated for 10 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50210048(CHEMBL3884919)
Affinity DataKi:  4.40E+4nMAssay Description:Inhibition of human LSD1 assessed as reduction in H2O2 production using H3K4me2 (1 to 20 residues) peptide as substrate preincubated for 10 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50210049(CHEMBL3885101)
Affinity DataKi:  1.90E+5nMAssay Description:Inhibition of human LSD1 assessed as reduction in H2O2 production using H3K4me2 (1 to 20 residues) peptide as substrate preincubated for 10 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50210050(CHEMBL3884529)
Affinity DataKi: >3.00E+5nMAssay Description:Inhibition of human LSD1 assessed as reduction in H2O2 production using H3K4me2 (1 to 20 residues) peptide as substrate preincubated for 10 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50210050(CHEMBL3884529)
Affinity DataKi: >3.00E+5nMAssay Description:Inhibition of human LSD1 assessed as reduction in H2O2 production using H3K4me2 (1 to 20 residues) peptide as substrate preincubated for 10 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed