Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 50048928
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of RIP1 (unknown origin) using MBP as substrate preincubated for 15 mins followed by MBP/ATP mixture addition measured after 90 mins by AD...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataIC50: 760nMAssay Description:Inhibition of recombinant GST-tagged RIP1 (unknown origin) after 4 hrs by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.50E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 262nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 198nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 64nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >5.00E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 1.08E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >3.00E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >3.00E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >3.00E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 490nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 1.23E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 656nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 8.24E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >3.00E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 98nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 628nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 378nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 2.53E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 221nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 1.74E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 1.25E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 36nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 627nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 815nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >3.00E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 1.23E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 72nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 457nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 898nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 4.10E+3nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Mouse)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 27nMAssay Description:Inhibition of RIP1 in mouse L929 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 6 hrs by Cell Titer-Glo luminescent cell vi...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
National Institute of Biological Sciences
Curated by ChEMBL
National Institute of Biological Sciences
Curated by ChEMBL
Affinity DataEC50: 74nMAssay Description:Inhibition of RIP1 in human HT-29 cells assessed as reduction in TNFalpha/z-VAD-FMK-induced necrosis after 24 hrs by Cell Titer-Glo luminescent cell ...More data for this Ligand-Target Pair