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Found 144 Enz. Inhib. hit(s) with all data for entry = 6070
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM67818(2-chloranyl-N-(3-quinoxalin-2-ylphenyl)ethanamide ...)
Affinity DataIC50:  0.200nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107139(US8592415, 24)
Affinity DataIC50:  0.300nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107142(US8592415, 27)
Affinity DataIC50:  0.600nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107137(US8592415, 22)
Affinity DataIC50:  45nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107124(US8592415, 8)
Affinity DataIC50:  136nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107125(US8592415, 9)
Affinity DataIC50:  175nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107131(US8592415, 16)
Affinity DataIC50:  270nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107136(US8592415, 21)
Affinity DataIC50:  330nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107133(US8592415, 18)
Affinity DataIC50:  500nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107120(US8592415, 4)
Affinity DataIC50:  2.70E+3nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107138(US8592415, 23)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107148(US8592415, 33)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107141(US8592415, 26)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107144(US8592415, 29)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107145(US8592415, 30)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107146(US8592415, 31)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107147(US8592415, 32)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107148(US8592415, 33)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107149(US8592415, 34)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107140(US8592415, 25)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107145(US8592415, 30)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107143(US8592415, 28)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107151(US8592415, 36)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107151(US8592415, 36)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107133(US8592415, 18)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107137(US8592415, 22)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107138(US8592415, 23)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107139(US8592415, 24)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107140(US8592415, 25)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107141(US8592415, 26)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107142(US8592415, 27)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107143(US8592415, 28)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107144(US8592415, 29)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107145(US8592415, 30)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107146(US8592415, 31)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107147(US8592415, 32)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107148(US8592415, 33)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107149(US8592415, 34)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107151(US8592415, 36)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107133(US8592415, 18)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107137(US8592415, 22)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107138(US8592415, 23)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107139(US8592415, 24)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107140(US8592415, 25)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107141(US8592415, 26)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107142(US8592415, 27)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107143(US8592415, 28)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107144(US8592415, 29)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107145(US8592415, 30)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Reaction Biology

US Patent
LigandPNGBDBM107146(US8592415, 31)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro kinase enzyme assay using Jak3, Jak2, Jak1, and Tyk2.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 144 total ) | Next | Last >>
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