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Found 2 Enz. Inhib. hit(s) with Target = '[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial' and Ligand = 'BDBM50529880'
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50529880(CHEMBL4579004)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of E2-activated human PDHK2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50529880(CHEMBL4579004)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of E2-activated human PDHK2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed