Found 3 Enz. Inhib. hit(s) with Target = '[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial' and Ligand = 'BDBM227594' Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Homo sapiens (Human))
Gwangju Institute of Science and Technology
Curated by ChEMBL
Gwangju Institute of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 760nMAssay Description:Inhibition of PDK4 (unknown origin)More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Homo sapiens (Human))
Gwangju Institute of Science and Technology
Curated by ChEMBL
Gwangju Institute of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 770nMpH: 7.5 T: 2°CAssay Description:To determine the IC50 for PDK inhibitors, a mixture containing 0.05-0.2 μM PDK, 6μM E1, with or without 0.5 μM of the PDC core E2/E3BP...More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Homo sapiens (Human))
Gwangju Institute of Science and Technology
Curated by ChEMBL
Gwangju Institute of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 840nMAssay Description:Inhibition of [3H]citalopram binding to serotonin transporter (SERT) of cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
