Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A' and Ligand = 'BDBM50130095'
Affinity DataKi: 19nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataEC50: 210nMAssay Description:Agonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as accumulation of IP1 incubated for 1 hr at 37 degC followed by 15 mins ...More data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Agonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as induction of intracellular calcium release measured for 90 secs by flu...More data for this Ligand-Target Pair