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Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A' and Ligand = 'BDBM50231640'
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50231640(CHEMBL285157 | TCMDC-123457)
Affinity DataKi:  125nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in HEK293 cell membranes measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50231640(CHEMBL285157 | TCMDC-123457)
Affinity DataIC50:  2.62E+3nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in CHOK1 cells assessed as inhibition of 5-HT induced inositol phosphate production incubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50231640(CHEMBL285157 | TCMDC-123457)
Affinity DataIC50:  2.63E+3nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in CHOK1 cells assessed as inhibition of 5-HT induced inositol phosphate production incubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed