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Report error Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A' and Ligand = 'BDBM50516998'
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50516998(CHEMBL4552542)
Affinity DataKi:  194nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in HEK293 cell membranes measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50516998(CHEMBL4552542)
Affinity DataIC50:  7.94E+3nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in CHOK1 cells assessed as inhibition of 5-HT induced inositol phosphate production incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50516998(CHEMBL4552542)
Affinity DataIC50:  7.98E+3nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in CHOK1 cells assessed as inhibition of 5-HT induced inositol phosphate production incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed