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Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 3A' and Ligand = 'BDBM50309861'
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50309861(4-(5-Methyloxazolo[4,5-b]pyridin-2-yl)-1,4-diazabi...)
Affinity DataKi:  269nMAssay Description:Displacement of [3H]LY278584 from mouse 5HT3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50309861(4-(5-Methyloxazolo[4,5-b]pyridin-2-yl)-1,4-diazabi...)
Affinity DataIC50:  5nMAssay Description:Agonist activity at human 5HT3 receptor expressed in human skin epithelial cells assessed as stimulation of calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed