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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50163460'
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM50163460(2-Amino-6-(2-hydroxy-ethylsulfanyl)-4-(3-trifluoro...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]DPCPX binding to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by PDSP Ki Database
LigandPNGBDBM50163460(2-Amino-6-(2-hydroxy-ethylsulfanyl)-4-(3-trifluoro...)
Affinity DataKi:  14.1nMAssay Description:Antagonist activity at adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed