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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50263180'
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50263180(CHEMBL4081224)
Affinity DataEC50:  38nMAssay Description:Inhibition of RIPK1 in mouse L929sA cells transfected with human Fas assessed as inhibition in TNF-induced necroptosis pretreated for 0.5 hrs followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50263180(CHEMBL4081224)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human A1AR expressed in FlpIn-CHO cells assessed as intracellular calcium mobilization by Fluo-4 dye-based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed