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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50415880'
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50415880(CHEMBL1097489)
Affinity DataKi:  15.8nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 60 mins by beta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50415880(CHEMBL1097489)
Affinity DataKi:  158nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NSCA-induced decrease in cAM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed