Report error Found 4 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a/A2b' and Ligand = 'BDBM50453223'
Affinity DataKi: 2.80nMAssay Description:Inhibition of adenylate cyclase via adenosine A1 receptors in rat fat cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatal membranes using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity against adenosine A2 receptor from human platelet membranes using [3H]NECAMore data for this Ligand-Target Pair
Affinity DataEC50: 414nMAssay Description:Maximal NECA stimulation of adenylate cyclase via adenosine A2 receptor in human platelet membranesMore data for this Ligand-Target Pair