TargetAdenosine receptor A2a(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universitat Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universitat Bonn
Curated by ChEMBL
Affinity DataKi: 3.79E+3nMAssay Description:Displacement of [3H]MSX-2 from recombinant human A2A adenosine receptor expressed in CHO cell membranes measured after 60 mins by liquid scintillatio...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Mus musculus)
Rheinische Friedrich-Wilhelms-Universitat Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universitat Bonn
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]MSX-2 from recombinant mouse A2A adenosine receptor expressed in CHO cell membranes measured after 60 mins by liquid scintillatio...More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+4nMAssay Description:Binding affinity for adenosine A2A receptor using [3H]-NECA in rat brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+4nMAssay Description:Displacement of [3H]NECA from rat A2A adenosine receptor expressed in CHO cell membranes measured after 60 mins by liquid scintillation counting meth...More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+4nMAssay Description:Displacement of [3H]R-PIA from adenosine A2A receptor in rat brain striatal membranesMore data for this Ligand-Target Pair