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Report error Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2b' and Ligand = 'BDBM50242058'
TargetAdenosine receptor A2b(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50242058(CHEMBL4070936)
Affinity DataKi:  1.80nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in HEK293 cells assessed as inhibition of NECA-induced increase in cAMP accumulation in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50242058(CHEMBL4070936)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Human)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50242058(CHEMBL4070936)
Affinity DataIC50:  2.00E+3nMAssay Description:Displacement of [3H]desmethoxy-verapamil from L-type calcium channel of bovine frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed