Report error Found 3 Enz. Inhib. hit(s) with Target = 'Aldo-keto reductase family 1 member B10' and Ligand = 'BDBM50362835'
Affinity DataKi: 2.60nMAssay Description:Competitive inhibition at human recombinant N-terminus His6-tagged AKR1B10 expressed in Escherichia coli BL21 DE3 assessed as inhibition of NADP+ lin...More data for this Ligand-Target Pair
Affinity DataIC50: 6.20nMAssay Description:Inhibition of human recombinant N-terminus His6-tagged AKR1B10 expressed in Escherichia coli BL21 DE3 assessed as pyridine-3-aldehyde reduction by sp...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of AKR1B10-mediated farnesal metabolism in human HeLa cells preincubated for 2 hrs measured after 6 hrs following [1-14C]farnesol additionMore data for this Ligand-Target Pair