Found 4 Enz. Inhib. hit(s) with Target = 'Alpha-1A adrenergic receptor' and Ligand = 'BDBM50421580' TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Affinity to Alpha-1 adrenergic receptor determined by radioligand binding techniques from rat-1 fibroblasts membranesMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:In vitro binding affinity against cloned human alpha-1A-adrenoreceptor receptors expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Activation of human alpha-1A adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Glaxosmithkline Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 4.60nMAssay Description:Agonist potency at Alpha-1A adrenoceptors assayed in rat-1 fibroblasts expressing human Alpha-1AMore data for this Ligand-Target Pair
