Report error Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-2A/Alpha-2B/Alpha-2C adrenergic receptor' and Ligand = 'BDBM50070100'
Affinity DataKi: 95nMAssay Description:Displacement of [3H]-RX-821002 from human alpha-2 adrenergic receptor in brain prefrontal cortex membrane by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataEC50: 4.23E+3nMAssay Description:Antagonist activity at human alpha-2 adrenergic receptor in brain prefrontal cortex membrane assessed as inhibition of UK14304-induced [35S]-GTPgamma...More data for this Ligand-Target Pair