Found 3 Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] A' and Ligand = 'BDBM19188'
Affinity DataKi: 1.57E+4nM ΔG°: -27.4kJ/molepH: 7.5 T: 2°CAssay Description:MAO A activities were determined spectrophotometrically at 316 nm using kynuramine as substrate. Competitive Ki values were determined by measuring i...More data for this Ligand-Target Pair
Affinity DataIC50: 5.89E+3nMAssay Description:Inhibition of Sprague-Dawley rat MAO-A using Kynuramine as substrate assessed as formation of 4-hydroxyquinoline preincubated for 5 mins prior to sub...More data for this Ligand-Target Pair
Affinity DataIC50: 5.94E+3nMAssay Description:Inhibition of MAO-A from Wistar rat brain by radioenzymatic assayMore data for this Ligand-Target Pair