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Found 2 Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] A' and Ligand = 'BDBM86776'
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM86776(Phthalonitrile analogue, 4e)
Affinity DataIC50:  399nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM86776(Phthalonitrile analogue, 4e)
Affinity DataIC50:  399nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed