BindingDB PrimarySearch

Found 5 Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] B' and Ligand = 'BDBM50049240'

Amine oxidase [flavin-containing] B(Homo sapiens (Human))
Dart Neuroscience

Curated by ChEMBL

BDBM50049240((+-)-5-((4-(2-(5-ethyl-2-pyridinyl)ethoxy)phenyl)m...)

Ki: 199nMAssay Description:Inhibition of human recombinant soluble MAO-B expressed in Pichia pastoris incubated for 30 mins prior to substrate addition measured after 60 mins b...More data for this Ligand-Target Pair

Amine oxidase [flavin-containing] B(Homo sapiens (Human))
Dart Neuroscience

Curated by ChEMBL

BDBM50049240((+-)-5-((4-(2-(5-ethyl-2-pyridinyl)ethoxy)phenyl)m...)

Ki: 271nMAssay Description:Inhibition of human recombinant microsomal MAO-B expressed in Pichia pastoris incubated for 30 mins prior to substrate addition measured after 60 min...More data for this Ligand-Target Pair

Amine oxidase [flavin-containing] B(Homo sapiens (Human))
Dart Neuroscience

Curated by ChEMBL

BDBM50049240((+-)-5-((4-(2-(5-ethyl-2-pyridinyl)ethoxy)phenyl)m...)

Ki: 500nMAssay Description:Competitive inhibition of human MAOB expressed in Pichia pastorisMore data for this Ligand-Target Pair

Amine oxidase [flavin-containing] B(Rattus norvegicus (rat))
TBA

Curated by ChEMBL

BDBM50049240((+-)-5-((4-(2-(5-ethyl-2-pyridinyl)ethoxy)phenyl)m...)

Ki: 2.10E+3nMAssay Description:Competitive inhibition of rat MAOB expressed in Pichia pastorisMore data for this Ligand-Target Pair

Amine oxidase [flavin-containing] B(Homo sapiens (Human))
Dart Neuroscience

Curated by ChEMBL

BDBM50049240((+-)-5-((4-(2-(5-ethyl-2-pyridinyl)ethoxy)phenyl)m...)

IC50: 298nMAssay Description:Inhibition of human recombinant MAO-B after 15 minsMore data for this Ligand-Target Pair