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Found 1 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM18195'
TargetAndrogen receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

LigandPNGBDBM18195(1-(2-methylpropyl)-9-(trifluoromethyl)-1H,2H,3H,6H...)
Affinity DataKi:  17nM ΔG°:  -46.1kJ/mole EC50:  3.20nMpH: 7.4 T: 2°CAssay Description:The compounds were evaluated in a transcriptional activation assay with hAR in a mammalian cell background (CV-1) as the primary in vitro assay. Rece...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed