Report error Found 6 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM493530'
Affinity DataKi: 3nMAssay Description:ReceptorsGR (human) (agonist radioligand) IM-9 cells (cytosol)[3H]dexamethasone 1.5 nM 1.5 nM triamcinolone (10 μM) 6 h 4° C. Scintillation coun...More data for this Ligand-Target Pair
Affinity DataIC50: 6.90nMAssay Description:ReceptorsGR (human) (agonist radioligand) IM-9 cells (cytosol)[3H]dexamethasone 1.5 nM 1.5 nM triamcinolone (10 μM) 6 h 4° C. Scintillation coun...More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Antagonist activity at Androgen receptor F877L mutant in human LNCaP cells measured by transcriptional reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Antagonist activity at AR F877L mutant (unknown origin) transfected in human LNCAP cells cotransfected with ARE-LUC incubated for 20 to 24 hrs in pre...More data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Antagonist activity at Androgen receptor in human LNCaP cells measured by transcriptional reporter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Antagonist activity at AR wild-type (unknown origin) transfected in human LNCAP cells cotransfected with ARE-LUC incubated for 20 to 24 hrs in presen...More data for this Ligand-Target Pair
