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Report error Found 2 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM50220941'
TargetAndrogen receptor(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50220941(5-(4-(4-((7R,8R,9S,10R,13S,14S,17S)-17-hydroxy-10,...)
Affinity DataIC50:  96nMAssay Description:Displacement of [3H]mibolerone from human androgen receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50220941(5-(4-(4-((7R,8R,9S,10R,13S,14S,17S)-17-hydroxy-10,...)
Affinity DataIC50:  250nMAssay Description:Antagonist activity at human androgen receptor expressed in HeLa cells assessed as inhibition of dihydrotestosterone induced transcriptional activity...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed