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Found 3 Enz. Inhib. hit(s) with Target = 'Apelin receptor' and Ligand = 'BDBM50577748'
TargetApelin receptor(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50577748(CHEMBL4870497)
Affinity DataEC50:  0.440nMAssay Description:Agonist activity at human APJ receptor expressed in HEK293T cells assessed as compound stimulated inhibition of forskolin stimulated cAMP production ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50577748(CHEMBL4870497)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at human APJ expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP production incubated for 60 mins by fluor...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetApelin receptor(Rattus norvegicus)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50577748(CHEMBL4870497)
Affinity DataEC50:  0.610nMAssay Description:Agonist activity at rat APJ receptor expressed in HEK293T cells assessed as compound stimulated inhibition of forskolin stimulated cAMP production in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed