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Found 4 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM50435003'
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University

Curated by ChEMBL
LigandPNGBDBM50435003(ENDOXIFEN)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human placental microsomal aromatase using testosterone as substrate assessed as formation of estradiol after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University

Curated by ChEMBL
LigandPNGBDBM50435003(ENDOXIFEN)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human recombinant placental aromataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University

Curated by ChEMBL
LigandPNGBDBM50435003(ENDOXIFEN)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluoresc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University

Curated by ChEMBL
LigandPNGBDBM50435003(ENDOXIFEN)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human aromatase assessed as reduction in fluorescence intensity preincubated with NADPH regenerating system for 10 mins followed by sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed