Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM9894'
TargetAromatase(Homo sapiens (Human))
Ohio State University

LigandPNGBDBM9894(2-(1H-Imidazol-1-yl)-3-(4-methoxyphenyl)-7-(benzyl...)
Affinity DataKi:  4.40E+3nM ΔG°:  -31.8kJ/mole IC50:  4.70E+3nMpH: 7.0 T: 2°CAssay Description:Inhibition of human placental aromatase was determined by monitoring the amount of 3H2O released as the enzyme converts [1beta-3H]androst-4-ene-3,17-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Ohio State University

LigandPNGBDBM9894(2-(1H-Imidazol-1-yl)-3-(4-methoxyphenyl)-7-(benzyl...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of human aromatase-mediated conversion of [1beta3H]androstenedione to estrone by liquid scintillation counting in presence of NADPHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed