TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 0.400nMAssay Description:Binding affinity at human adrenergic beta2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 0.537nMAssay Description:Displacement of [3H]-CGP 12177 from human beta-2 adrenergic receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.661nMAssay Description:Antagonist activity at human beta-2 adrenergic receptor expressed in salbutamol-stimulated CHO-K1 cells assessed as CRE-SPAP level by fluorescence co...More data for this Ligand-Target Pair