Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Bile acid receptor' and Ligand = 'BDBM50090940'
TargetBile acid receptor(Homo sapiens (Human))
Glaxo Wellcome Research & Development

Curated by ChEMBL
LigandPNGBDBM50090940(3-(2-{4-[3-(2,6-Dichloro-phenyl)-5-methyl-isoxazol...)
Affinity DataEC50:  70nMAssay Description:Ligand dependent recruitment of SRC1(676-700) peptide to human Farnesoid X-activated receptor by fluorescence resonance energy transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Glaxo Wellcome Research & Development

Curated by ChEMBL
LigandPNGBDBM50090940(3-(2-{4-[3-(2,6-Dichloro-phenyl)-5-methyl-isoxazol...)
Affinity DataEC50:  4.10E+3nMAssay Description:Agonist activity at FXR (unknown origin) by cell based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Glaxo Wellcome Research & Development

Curated by ChEMBL
LigandPNGBDBM50090940(3-(2-{4-[3-(2,6-Dichloro-phenyl)-5-methyl-isoxazol...)
Affinity DataEC50:  70nMAssay Description:Agonist activity at FXR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed