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Report error Found 2 Enz. Inhib. hit(s) with Target = 'Bile acid receptor' and Ligand = 'BDBM50258557'
TargetBile acid receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50258557(3-(2-chloro-4-((3-(2,6-dichlorophenyl)-5-(pentan-3...)
Affinity DataEC50:  280nMAssay Description:Agonist activity at human FXR assessed as SRC1 coactivatior peptide recruitment by cell free FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile acid receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50258557(3-(2-chloro-4-((3-(2,6-dichlorophenyl)-5-(pentan-3...)
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist activity at human FXR assessed as SRC1 peptide interaction with receptor ligand binding domain by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed