Found 1 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 1' and Ligand = 'BDBM50558065'
TargetBromodomain-containing protein 1(Homo sapiens (Human))
Constellation Pharmaceuticals
Curated by ChEMBL
Constellation Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.50E+4nMAssay Description:Inhibition of BRD1 (unknown origin) measured after 70 mins by TR-FRET assayMore data for this Ligand-Target Pair