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Found 3 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 3' and Ligand = 'BDBM50543359'
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50543359(GSK620)
Affinity DataIC50:  72nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) assessed as dissociation constant by TR-FRET methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50543359(GSK620)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of BRD3-BD1 (unknown origin) assessed as dissociation constant by TR-FRET methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50543359(GSK620)
Affinity DataIC50:  2.51E+4nMAssay Description:Binding affinity to 6His-Thr-BRD3 (1 to 435 residues) BD1 domain (unknown origin) incubated for 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed