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Found 4 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 3' and Ligand = 'BDBM50544300'
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50544300(GSK046)
Affinity DataIC50:  98nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) assessed as dissociation constant by TR-FRET methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50544300(GSK046)
Affinity DataIC50:  100nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from 6His-Thr tagged BRD3 BD2/BD1 Y73A mutant (1 to 435 residues) (unknown origin) measured after 30 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50544300(GSK046)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of BRD3-BD1 (unknown origin) assessed as dissociation constant by TR-FRET methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50544300(GSK046)
Affinity DataIC50:  3.98E+4nMAssay Description:Displacement of Alexa Fluor 647 labelled ligand from 6His-Thr tagged BRD3 BD1/BD2 Y348A mutant (1 to 435 residues) (unknown origin) measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed