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Found 6 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM50463897'
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)
Affinity DataIC50:  15nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 4 hrs by alpha-screen as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)
Affinity DataIC50:  50nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)
Affinity DataIC50:  50nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)
Affinity DataIC50:  60nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1/BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-scr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)
Affinity DataIC50:  75nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 1 hr by alpha-screen ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)
Affinity DataIC50:  274nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 5 mins by alpha-screen a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed