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Found 3 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM50586215'
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586215(CHEMBL5080392)
Affinity DataIC50:  775nMAssay Description:Binding affinity to human partial length BRD4-BD2 (K333 to E460 residues) expressed in bacterial system assessed as dissociation constant by BROMOsca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586215(CHEMBL5080392)
Affinity DataIC50:  900nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Cnrs

Curated by ChEMBL
LigandPNGBDBM50586215(CHEMBL5080392)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 6 hrs by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed